Green, catalyst-free synthesis of mesalazine conjugates

Mohamed A. Ibrahim, Siva S. Panda, Khalid A. Alamry, Alan R. Katritzky

Research output: Contribution to journalArticle

1 Citation (Scopus)

Abstract

A greener protocol for the synthesis of mesalazine conjugates is reported. Mesalazine conjugates are prepared in high yields by a one-pot reaction of mesalazine and aminoacyl/peptidoylbenzotriazoles in water under microwave irradiation.

Original languageEnglish (US)
Pages (from-to)3255-3258
Number of pages4
JournalSynthesis (Germany)
Volume45
Issue number23
DOIs
StatePublished - 2013

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Mesalamine
Microwave irradiation
Catalysts
Water

Keywords

  • amino acid
  • benzotriazole methodology
  • green chemistry
  • mesalazine
  • prodrug

ASJC Scopus subject areas

  • Organic Chemistry
  • Catalysis

Cite this

Green, catalyst-free synthesis of mesalazine conjugates. / Ibrahim, Mohamed A.; Panda, Siva S.; Alamry, Khalid A.; Katritzky, Alan R.

In: Synthesis (Germany), Vol. 45, No. 23, 2013, p. 3255-3258.

Research output: Contribution to journalArticle

Ibrahim, MA, Panda, SS, Alamry, KA & Katritzky, AR 2013, 'Green, catalyst-free synthesis of mesalazine conjugates', Synthesis (Germany), vol. 45, no. 23, pp. 3255-3258. https://doi.org/10.1055/s-0033-1338532
Ibrahim, Mohamed A. ; Panda, Siva S. ; Alamry, Khalid A. ; Katritzky, Alan R. / Green, catalyst-free synthesis of mesalazine conjugates. In: Synthesis (Germany). 2013 ; Vol. 45, No. 23. pp. 3255-3258.
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